For a deeper dive

Compact hydrophilic electrophiles enable highly efficacious high DAR ADCs with excellent in vivo PK profile Chemical Science 2023

Targeting FLT3 By New-Generation Antibody-Drug-Conjugate In Combination With KinaseInhibitors For Treatment Of AML. Blood 2022

Bis-ethynyl-phosphonamidatesas an Modular Conjugation Platform to Generate Multifunctional Protein- and Antibody-Drug-Conjugates. European Journal of Organic Chemistry 2022

Ethynyl-phosphonamidates for the Rapid and Cysteine-Selective Generation of Efficacious Antibody-Drug Conjugates. Angewandte Chemie 2019

Cysteine-Selective Phosphonamidate Electrophiles for Modular Protein Bioconjugations. Angewandte Chemie 2019

Versatile and Efficient Site-Specific Protein Functionalization by Tubulin Tyrosine Ligase. Angewandte Chemie 2015